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Class Explorer · Anti-infectives

Nitroimidazoles

Reduced inside anaerobic organisms to radicals that fragment DNA. The reduction only happens in a low-oxygen environment, which is the entire basis of the spectrum.

Members

Also in this class: Tinidazole. Full pages arrive as the library grows.

Compare the members

Metronidazole
Spectrum
Anaerobes and protozoa
Counselling
No alcohol during, and 48 h after

Shared across the class

Indications
Anaerobic infection · C. difficile (no longer first line) · Bacterial vaginosis, trichomoniasis, giardiasis, amoebiasis · Intra-abdominal infection as part of combination therapy
Adverse effects
Metallic taste · Nausea · Peripheral neuropathy on prolonged use · Disulfiram-like reaction with alcohol
Contraindications
First trimester of pregnancy, relative · Alcohol during and for 48 hours after
Monitoring
Neuropathy symptoms on courses beyond a few weeks · Alcohol counselling, which has to be explicit

What makes each agent different

  • Tinidazole has a longer half-life allowing shorter courses; the spectrum is essentially the same.

It has no aerobic Gram-negative activity at all, so it is a partner drug in intra-abdominal sepsis, never a solo one.

The alcohol reaction is often dismissed as folklore; it is unpleasant enough that the warning belongs on the label and in the conversation.

Last reviewed 2026-08-16 · Goodman & Gilman's The Pharmacological Basis of Therapeutics, 14th ed.