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Opioids · Pain & inflammation

Oxycodone

OxyNEO® · Percocet (with acetaminophen)®(brand names vary by market)

Reliable oral absorption, and a combination product that hides a second drug.

Illustration of Oxycodone as a tabletOXY

Also: modified release, oral liquid

Mechanism

Mu opioid receptor agonist with higher and more predictable oral bioavailability than morphine.

Indications

  • Moderate to severe pain
  • Post-operative pain
  • Cancer pain

Formulations

TabletModified releaseOral liquid

Dosing concepts

Combination products

Frequently combined with acetaminophen, which places a hard ceiling on the dose that has nothing to do with the opioid. Escalating the opioid then risks hepatotoxicity from the other half.

Modified release

Long-acting forms are for stable background pain, never for acute or breakthrough use, and are swallowed whole.

Concepts, not prescribing instructions. Practice numbers live in current references and local protocols.

Pharmacokinetics

Bioavailability
~60 to 87%, the highest of the common oral opioids
Half-life
3 to 5 h
Elimination
hepatic: CYP3A4 and CYP2D6; strong CYP3A4 inhibitors raise exposure
Protein binding
~45%
Play with these concepts in the PK Lab

Adverse effects

  • Constipationcommon
  • Sedationcommon & serious
  • Nauseacommon
  • Respiratory depressionserious
  • Dependence and use disorderseriousIts abuse liability is a matter of public record and shapes how it is prescribed.

Contraindications & precautions

Contraindications

  • Respiratory depression
  • Paralytic ileus
  • Acute severe asthma without support

Precautions

  • Combination products containing acetaminophen
  • Concurrent CYP3A4 inhibitors
  • History of substance use disorder

Interactions

Monitoring

Total acetaminophen dose from all sources

The combination product is a hidden acetaminophen prescription

Sedation and bowel function

Class effects

Duration and quantity supplied

Prescribing practice is itself a safety intervention here

Counselling points

  • If your tablets contain acetaminophen as well, do not take any other product containing it.
  • Swallow long-acting tablets whole.
  • Take a laxative regularly.
  • Keep it locked away and return unused tablets to a pharmacy.

Clinical pearls

  • Combination oxycodone-acetaminophen tablets are a leading route to accidental acetaminophen overdose, because the patient counts opioid tablets and adds a separate acetaminophen on top.
  • Its high oral bioavailability makes the oral route genuinely reliable, which is a real advantage over morphine outside hospital.

References & review

  • Oxycodone product monograph (consult the current version for your market) (monograph)
  • Goodman & Gilman's The Pharmacological Basis of Therapeutics, 14th ed. (reference-work)

Last reviewed 2026-08-16 · jurisdiction: global · drug information changes; verify against current references before practice use.